TIANEPTINE SODIUM LIQUID SOLUTION.
25mg/mL – 30mL Bottle.
Buy Tianeptine Sodium Liquid Solution. [>99.8% Purity]. Water Soluble.
Inactive Ingredients: Solvent Matrix. Preservative.
Tianeptine was developed in France in the 1960’s.
Tianeptine’s mechanism of action is not fully understood. Research shows that it possesses SSRE (selective serotonin reuptake enhancer) properties, which is very different than the popular SSRI (selective serotonin reuptake inhibitor) compounds. Both serotonin re-uptake enhancement and serotonin re-uptake inhibition takes place via the compounds modulating the serotonin transporter (SERT). One of the other noteworthy effects of Tianeptine is its ability to inhibit glutaminergic (excitatory) neurotransmission by modulating the AMPA and NMDA receptors, which has shown to mitigate stress-induced unfavorable changes in neurotransmitter balance. It is believed that these effects are also why Tianeptine has shown to promote neural plasticity in some studies, partly via elevations in BDNF (brain-derived neurotrophic factor). Furthermore, Tianpetine exerts a mild agonist (activating) effect at the μ-opioid receptor (MOR), based on available data.
Tianeptine sodium has the highest bio-availability and most rapid onset, compared to other forms of Tianeptine. Tianeptine sodium shows a bio-availability of ~99%, with primary metabolism being hepatic (liver), and a half-life of 2-3 hours.
Buy Tianeptine from ELV Bioscience.
This product is for laboratory use and research purposes only.
CONTACT US for bulk quantities.